SCHEMBL9809398

SCHEMBL9809398

O=C(O)CC(O)(SCc1ccccc1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.44
AKR1B1 P15121 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
SLC13A5 Q86YT5 2/20 0.41
CYP3A4 P08684 1/20 0.41
PRMT1 Q99873 1/20 0.41
PAM P19021 1/20 0.41
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
HIF1A Q16665 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KEAP1 Q14145 1/20 0.38
FFAR1 O14842 2/20 0.37
IDO1 P14902 2/20 0.37
MMP12 P39900 1/20 0.37
MMP13 P45452 1/20 0.37
CES2 O00748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10404926 0.84 SLC13A5 (0.46) CYP2C19AKR1B1CYP1A2CYP2D6SLC13A5
SCHEMBL6431176 0.76 CYP3A4 (0.59) CYP2C19AKR1B1CYP1A2CYP2D6CYP3A4
SCHEMBL3347786 0.74 GAA (0.43) MEN1KMT2A
SCHEMBL10630052 0.74 CYP2C19 (0.43) CYP2C19AKR1B1CYP1A2CYP2D6CYP3A4
SCHEMBL27862577 0.72 CYP2C19 (0.53) CYP2C19AKR1B1CYP1A2CYP2D6CYP3A4
SCHEMBL10824526 0.72 ALDH1A1 (0.46) CYP2C19CYP2D6HIF1AADRA1A
SCHEMBL9068773 0.72 CYP1A2 (0.53) CYP2C19AKR1B1CYP1A2CYP2D6CYP3A4
SCHEMBL1952401 0.71 CYP2C19 (0.47) CYP2C19CYP1A2SLC13A5HIF1AKEAP1
Propionic Acid SCHEMBL11592770 0.70 CYP1A2 (0.47) CYP2C19AKR1B1CYP1A2CYP2D6CYP3A4
SCHEMBL499117 0.69 CYP2C19 (0.64) CYP2C19AKR1B1CYP1A2PAMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4985485-A HYDROTALCITE RHONE-POULENC CHIMIE (FR) 1991-01-15 US disclosed
US-4963594-A STABILIZERS OF THIOMALIC ACID DIESTERS, ZINC AND GROUP IIA CARBOXYLIC ACID SALTS AND PHENOLATES; MOLDING MATERIALS, COLORFAST RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1990-10-16 US disclosed
US-4921896-A RED PHOSPHORUS, LANTHANIDE, TALC, ZINC SULFIDE OR ZINC OXIDE RHONE-POULENC CHIMIE (FR) 1990-05-01 US disclosed
US-4612339-A YTTRIUM OR LANTHANDIDE COMPOUND; AMMONIUM, ALKALI OR ALKALINE EARTH METAL HALIDE RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1986-09-16 US disclosed
US-4559372-A ADDITIVES OF RED PHOSPHORUS AND A LANTHANIDE AND/OR YTTRIUM COMPOUND; NONTOXIC;ARC TRACKING RESISTANCE RHONE-POULENC SPECIALITIES CHIMIQUES (FR) 1985-12-17 US disclosed