SCHEMBL981182

SCHEMBL981182

O=C(CN1CCNCC1)NC1CCC(O)CC1

nearest known ligand 0.74

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.74
CHRM5 P08912 4/20 0.74
CHRM3 P20309 3/20 0.74
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA9 Q16790 2/20 0.46
EPHX2 P34913 1/20 0.44
PKM P14618 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
SMYD3 Q9H7B4 1/20 0.41
CHRM1 P11229 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1901358 0.93 SIGMAR1 (0.84) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL982065 0.87 SIGMAR1 (0.90) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL11627783 0.86 SIGMAR1 (0.72) SIGMAR1CHRM5CHRM3CA12CA1
Esaprazole SCHEMBL931007 0.85 SIGMAR1 (1.00) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL976514 0.83 SIGMAR1 (0.68) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL13640016 0.83 SIGMAR1 (0.72) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL28391152 0.83 SIGMAR1 (0.72) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL1073695 0.83 SIGMAR1 (0.82) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL976989 0.82 SIGMAR1 (0.67) SIGMAR1CHRM5CHRM3CA12CA1
SCHEMBL12814299 0.81 SIGMAR1 (0.71) SIGMAR1CHRM5CHRM3CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011000945-A9 AMINOALKAMIDES FOR USE IN THE TREATMENT OF INFLAMMATORY, DEGENERATIVE OR DEMYELINATING DISEASES OF THE CNS NENSIUS RESEARCH A/S (DK) 2011-04-07 WO disclosed
WO-2011000945-A2 AMINOALKAMIDES FOR USE IN THE TREATMENT OF INFLAMMATORY, DEGENERATIVE OR DEMYELINATING DISEASES OF THE CNS NENSIUS RESEARCH A/S (DK) 2011-01-06 WO disclosed