SCHEMBL9811865

SCHEMBL9811865

CS(=O)(=O)Nc1ccc(NC(=S)C(P(=O)(O)O)P(=O)(O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.48
LMNA P02545 3/20 0.48
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
KEAP1 Q14145 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
XDH P47989 1/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KIF11 P52732 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CSNK2A1 P68400 1/20 0.39
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9435877 0.85 ALDH1A1 (0.49) KDM4EALDH1A1HPGDSMN1; SMN2KEAP1
SCHEMBL10412485 0.82 KDM4E (0.44) KDM4ELMNAALDH1A1HPGDHTT
SCHEMBL9811856 0.80 CA12 (0.53) LMNAHPGDHTTSMN1; SMN2CA12
SCHEMBL9811848 0.79 SMN1; SMN2 (0.50) KDM4EALDH1A1HPGDHTTSMN1; SMN2
SCHEMBL9435834 0.77 KDM4E (0.46) KDM4EALDH1A1CA2CA9NPSR1
SCHEMBL9811859 0.77 CA12 (0.53) LMNAALDH1A1SMN1; SMN2CA12CA1
SCHEMBL233680 0.76 CA9 (0.50) KDM4ELMNAALDH1A1SMN1; SMN2CA12
SCHEMBL9811871 0.76 IDO1 (0.50) KDM4ELMNAALDH1A1HPGDSMN1; SMN2
SCHEMBL9811870 0.73 CA12 (0.57) CA12CA1KIF11TRPV1
SCHEMBL12421869 0.71 KEAP1 (0.52) KDM4ELMNAALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0243173-B1 NEW DIPHOSPHONIC ACID COMPOUNDS, PROCESSES FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-06-26 EP disclosed
US-4963536-A INHIBIT BONE RESORPTION FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1990-10-16 US disclosed
US-4857513-A Diphosphonic acid compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISIWA PHARMACEUTICAL CO., LTD. (JP) 1989-08-15 US disclosed
EP-0243173-A2 New diphosphonic acid compounds, processes for the preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-10-28 EP disclosed