SCHEMBL9813193

SCHEMBL9813193

COc1ccc2c(c1)[S+]([O-])c1cc(OC(C)=O)c(OC)cc1N2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNFSF11 O14788 1/20 0.42
BACE1 P56817 1/20 0.42
TSHR P16473 3/20 0.39
JUN P05412 1/20 0.39
NFKB1 P19838 1/20 0.39
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38
TUBB6 Q9BUF5 1/20 0.38
TUBB2B Q9BVA1 1/20 0.38
TUBB1 Q9H4B7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9813221 0.79 TUBB4A (0.41) BACE1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9813149 0.76 SNCA (0.61) TNFSF11BACE1TSHRTUBB4ATUBB
SCHEMBL9813220 0.75 KMT2A (0.58) TNFSF11BACE1TSHRTUBB4ATUBB
SCHEMBL3328971 0.71 TSHR (0.64) TNFSF11BACE1TSHRJUNNFKB1
SCHEMBL3327344 0.71 CA12 (0.63) TNFSF11BACE1TSHRTUBB4ATUBB
SCHEMBL11793587 0.70 BACE1 (0.61) TNFSF11BACE1TSHRJUNNFKB1
SCHEMBL20551035 0.68 NOX1 (0.50) MEN1KMT2AALDH1A1MAPTL3MBTL1
SCHEMBL21723164 0.67 TNFSF11 (0.83) TNFSF11BACE1TSHRJUNNFKB1
SCHEMBL27602532 0.67 TNFSF11 (0.83) TNFSF11BACE1TSHRJUNNFKB1
SCHEMBL8928654 0.67 TNFSF11 (0.83) TNFSF11BACE1TSHRJUNNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0138481-B1 LEUKOTRIENE BIOSYNTHESIS INHIBITORS MERCK FROSST CANADA INC. (CA) 1991-06-26 EP disclosed
US-4845083-A PHENOTHIAZINE DERIVATIVES AND ANALOGS MERCK FROSST CANADA, INC. (CA) 1989-07-04 US disclosed
EP-0138481-A2 Leukotriene biosynthesis inhibitors MERCK FROSST CANADA INC. (CA) 1985-04-24 EP disclosed