SCHEMBL98136

SCHEMBL98136

COc1ccc(Sc2nc(N3CCOCC3)c3ncn(CC4CC4)c3n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 5/20 0.43
MTOR P42345 3/20 0.43
PIK3CG P48736 3/20 0.43
ATR Q13535 2/20 0.42
NOS1 P29475 1/20 0.41
CNR2 P34972 3/20 0.40
PDE10A Q9Y233 2/20 0.39
TLR9 Q9NR96 3/20 0.39
TLR7 Q9NYK1 2/20 0.39
MERTK Q12866 1/20 0.38
HDAC1 Q13547 3/20 0.37
PIK3R1 P27986 2/20 0.37
STAT3 P40763 1/20 0.37
ATRIP Q8WXE1 1/20 0.37
PIK3CD O00329 1/20 0.37
PIK3CB P42338 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL98137 0.87 ALDH1A1 (0.49) PIK3CAMTORPIK3CGATRNOS1
SCHEMBL99029 0.78 ALDH1A1 (0.49) PIK3CAMTORPIK3CGNOS1CNR2
SCHEMBL30440406 0.74 PIK3CA (0.52) PIK3CAMTORPIK3CGATRCNR2
SCHEMBL336380 0.74 PIK3CA (0.52) PIK3CAMTORPIK3CGATRCNR2
SCHEMBL98344 0.73 ALDH1A1 (0.49) PIK3CANOS1CNR2PDE10ATLR9
SCHEMBL100676 0.73 ALDH1A1 (0.49) PIK3CANOS1CNR2PDE10ATLR9
SCHEMBL98831 0.72 PDE10A (0.41) PIK3CAATRNOS1PDE10AMERTK
SCHEMBL99742 0.71 PIK3CA (0.37) PIK3CANOS1CNR2PDE10ATLR9
SCHEMBL98381 0.71 ALDH1A1 (0.54) PIK3CANOS1PDE10ATLR9TLR7
SCHEMBL336204 0.71 PIK3CA (0.67) PIK3CAMTORPIK3CGHDAC1PIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-B1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KK (JP) 2015-03-11 EP disclosed
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed