SCHEMBL99742

SCHEMBL99742

CCOC1CN(c2nc(Sc3ccc(OC)cc3)nc3c2ncn3C)CCO1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.37
CNR2 P34972 2/20 0.37
FFAR2 O15552 2/20 0.34
CCNE2 O96020 2/20 0.33
CCNE1 P24864 2/20 0.33
CDK2 P24941 2/20 0.33
SRC P12931 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
TLR9 Q9NR96 4/20 0.33
TLR7 Q9NYK1 3/20 0.33
PDE10A Q9Y233 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
HSP90B1 P14625 1/20 0.32
NOS1 P29475 1/20 0.32
ADORA1 P30542 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99741 0.88 ALDH1A1 (0.41) PIK3CACNR2FFAR2CCNE2CCNE1
SCHEMBL99474 0.79 PIK3CA (0.35) PIK3CACNR2SRC
SCHEMBL99160 0.78 ALDH1A1 (0.38) PIK3CAFFAR2
SCHEMBL1674720 0.76 PIK3CA (0.31) PIK3CA
SCHEMBL98898 0.76 GSK3B (0.35) PIK3CA
SCHEMBL97904 0.75 ALDH1A1 (0.44)
SCHEMBL98824 0.74 ALDH1A1 (0.40) PIK3CACNR2SRCPDE10A
SCHEMBL1620825 0.73 ALDH1A1 (0.33) PIK3CASRC
SCHEMBL98136 0.71 PIK3CA (0.43) PIK3CACNR2TLR9TLR7PDE10A
SCHEMBL100748 0.71 CNR2 (0.35) PIK3CACNR2SRCTLR9TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426130-B1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KK (JP) 2015-03-11 EP disclosed
EP-2426130-A1 PURINE DERIVATIVE AND ANTITUMOR AGENT USING SAME ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 2012-03-07 EP disclosed