SCHEMBL9813896

SCHEMBL9813896

Oc1ccc(CCN(CC(O)c2ccccc2)C[C@H](O)c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 8/20 0.51
OPRM1 P35372 7/20 0.51
OPRD1 P41143 7/20 0.51
KDM4E B2RXH2 3/20 0.47
TAAR1 Q96RJ0 1/20 0.46
CYP51A1 Q16850 2/20 0.45
AOC3 Q16853 2/20 0.45
RET P07949 1/20 0.44
KDR P35968 1/20 0.44
BCHE P06276 1/20 0.43
ALDH1A1 P00352 1/20 0.42
GLI1 P08151 1/20 0.42
GLI2 P10070 1/20 0.42
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10339989 0.83 SLC2A1 (0.46) OPRK1OPRM1OPRD1CYP51A1
SCHEMBL9813954 0.83 SLC2A1 (0.46) OPRK1OPRM1OPRD1CYP51A1
SCHEMBL9813931 0.83 SLC2A1 (0.46) OPRK1OPRM1OPRD1CYP51A1
SCHEMBL9813927 0.83 OPRK1 (0.42) OPRK1OPRM1OPRD1CYP51A1
Hydrochloric Acid SCHEMBL11479900 0.83 ADRA2A (0.54) OPRM1KDM4ETAAR1AOC3BCHE
SCHEMBL4479037 0.82 GLI1 (0.50) OPRK1OPRM1OPRD1KDM4ETAAR1
SCHEMBL4479042 0.82 GLI1 (0.50) OPRK1OPRM1OPRD1KDM4ETAAR1
SCHEMBL10822409 0.81 KDM4E (0.50) OPRK1OPRM1OPRD1KDM4ETAAR1
SCHEMBL10822410 0.81 KDM4E (0.50) OPRK1OPRM1OPRD1KDM4ETAAR1
SCHEMBL10822407 0.81 KDM4E (0.50) OPRK1OPRM1OPRD1KDM4ETAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017619-A Anitdiabetic HOFFMANN-LA ROCHE INC. (US) 1991-05-21 US disclosed
EP-0198412-B1 PHENETHANOL AMINE DERIVATIVES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1989-03-22 EP disclosed
EP-0198412-A1 Phenethanol amine derivatives F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1986-10-22 EP disclosed