SCHEMBL9815609

SCHEMBL9815609

COc1ccc(CCN(C)CC(C#N)=Cc2cc(CN3CCOCC3)c(O)c(OC)c2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
MAPT P10636 5/20 0.40
LMNA P02545 3/20 0.40
GAA P10253 3/20 0.40
MAPK1 P28482 3/20 0.40
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EGFR P00533 2/20 0.38
ERBB2 P04626 2/20 0.38
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9815602 0.88 MEN1 (0.46) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL9815632 0.84 CYP3A4 (0.54) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL9815610 0.81 MEN1 (0.44) MEN1KMT2AMAPTLMNAGAA
SCHEMBL9815622 0.73 CYP3A4 (0.48) MEN1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL11758665 0.72 NPC1 (0.52) MEN1KMT2ACYP1A2MAPTKDM4E
SCHEMBL9813043 0.71 GAA (0.52) MEN1KMT2ACYP3A4CYP2D6MAPT
SCHEMBL9815604 0.70 MEN1 (0.45) MEN1KMT2AMAPK1KDM4EALDH1A1
SCHEMBL3103923 0.70 GAA (0.53) MEN1KMT2AMAPTLMNAGAA
SCHEMBL11762690 0.67 KMT2A (0.56) MEN1KMT2AMAPTLMNAMAPK1
SCHEMBL11759526 0.67 ALDH1A1 (0.49) MEN1KMT2AMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266549-B1 CINNAMYL AMINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1991-06-19 EP disclosed