SCHEMBL9815982

SCHEMBL9815982

COc1ccccc1N1CCN(CC(O)COc2ccc(C(=CN(C)C)C(C)=O)cc2)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.61
CACNA1G O43497 1/20 0.61
ABCB1 P08183 7/20 0.58
HTR7 P34969 1/20 0.58
MAPT P10636 5/20 0.57
ALDH1A1 P00352 2/20 0.57
LMNA P02545 5/20 0.56
MAPK1 P28482 3/20 0.56
HTT P42858 1/20 0.56
HSP90AB1 P08238 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.55
TDP1 Q9NUW8 2/20 0.55
NR1I2 O75469 1/20 0.55
NR3C1 P04150 1/20 0.55
ADRB1 P08588 1/20 0.55
HTR1A P08908 1/20 0.55
ADRA2A P08913 1/20 0.55
DRD2 P14416 1/20 0.55
ADRA2B P18089 1/20 0.55
ADRA2C P18825 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9815989 0.91 ABCB1 (0.60) KCNH2CACNA1GABCB1MAPTALDH1A1
SCHEMBL9815959 0.89 ABCB1 (0.74) ABCB1HTR7
SCHEMBL10839674 0.86 HTR7 (0.73) ABCB1HTR7MAPTALDH1A1LMNA
SCHEMBL10837921 0.84 CACNA1G (0.65) KCNH2CACNA1GABCB1HTR7MAPT
SCHEMBL9815996 0.83 ABCB1 (0.61) ABCB1MEN1KMT2A
Hydrochloric Acid SCHEMBL11491672 0.81 CACNA1G (0.60) KCNH2CACNA1GABCB1MAPTALDH1A1
SCHEMBL30383961 0.81 KCNH2 (0.61) KCNH2CACNA1GABCB1HTR7MAPT
SCHEMBL3440691 0.81 KCNH2 (0.61) KCNH2CACNA1GABCB1HTR7MAPT
SCHEMBL3440692 0.81 KCNH2 (0.61) KCNH2CACNA1GABCB1HTR7MAPT
SCHEMBL17313697 0.81 KCNH2 (0.78) KCNH2CACNA1GABCB1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0167121-B1 SUBSTITUTED PHENYLPIPERAZINYL PROPANOLS, PROCESS FOR THEIR PREPARATION, THEIR USE, AND COMPOSITIONS CONTAINING THESE COMPOUNDS Beiersdorf Aktiengesellschaft (DE) 1991-10-23 EP disclosed
US-4631281-A ANTICOAGULANTS, ASTHMA, HYPOTENSIVE AGENTS, BRONCHOPILATORS, INOTROPIC AGENTS BEIERSDORF AKTIENGESELLSCHAFT (DE) 1986-12-23 US disclosed
EP-0167121-A2 Substituted phenylpiperazinyl propanols, process for their preparation, their use, and compositions containing these compounds Beiersdorf Aktiengesellschaft (DE) 1986-01-08 EP disclosed