SCHEMBL9816657

SCHEMBL9816657

C=CCNC(=O)/C=C(/C)N

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.45
ALDH1A1 P00352 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.39
FAAH O00519 1/20 0.39
RAB9A P51151 3/20 0.38
NPC1 O15118 1/20 0.38
KDM4E B2RXH2 1/20 0.37
PKM P14618 1/20 0.35
HPGD P15428 3/20 0.33
MAPK1 P28482 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9816659 1.00 TSHR (0.45) TSHRALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL4205555 0.83 SMN1; SMN2 (0.45) TSHRALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL11049989 0.78 ALDH1A1 (0.40) TSHRALDH1A1SMN1; SMN2MAPTKDM4E
SCHEMBL15482579 0.78 KMT2A (0.42) TSHRALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL15780411 0.76
SCHEMBL15482637 0.75 SMN1; SMN2 (0.38) TSHRALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL15482567 0.75 FAAH (0.47) TSHRALDH1A1SMN1; SMN2MAPTKMT2A
Acrylamide SCHEMBL9362700 0.74 ALDH1A1 (0.52) TSHRALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL11052618 0.74 KDM4E (0.46) ALDH1A1SMN1; SMN2MAPTKMT2AKDM4E
Butanedione SCHEMBL27637216 0.74 ALDH1A1 (0.48) TSHRALDH1A1SMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220653-B1 3-AMINOCARBONYL-1,4-DIHYDROPYRIDINE-5-CARBOXYLIC ACID COMPOUNDS, PROCESS FOR PREPARATION AND USE THEREOF, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Nippon Shoji Kabushiki Kaisha (JP) 1991-11-06 EP disclosed
US-4874773-A HYPOTENSIVE AGENTS, VASODILATORS NIPPON SHOJI KABUSHIKI KAISHA (JP) 1989-10-17 US disclosed
EP-0220653-A2 3-Aminocarbonyl-1,4-dihydropyridine-5-carboxylic acid compounds, process for preparation and use thereof, and pharmaceutical composition containing the same Nippon Shoji Kabushiki Kaisha (JP) 1987-05-06 EP disclosed