SCHEMBL9817664

SCHEMBL9817664

CCOC(=O)Cc1ccccc1C#Cc1ccc2c(c1)C(SC)(SC)CCO2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.35
S1PR5 Q9H228 2/20 0.33
CASP3 P42574 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
RAB9A P51151 1/20 0.33
FFAR1 O14842 1/20 0.32
CYP3A4 P08684 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
KMT2A Q03164 1/20 0.32
LMNA P02545 1/20 0.32
CNR2 P34972 1/20 0.32
PRSS1 P07477 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817771 0.91 CYP4F2 (0.39) S1PR5CASP3SENP8SENP7SENP6
SCHEMBL9817696 0.90 CYP4F2 (0.38) S1PR5FFAR1CYP3A4
SCHEMBL9817635 0.89 CYP4F2 (0.41) S1PR5FFAR1CYP3A4
SCHEMBL9817731 0.88 RARA (0.39) HPGDS1PR5CASP3SENP8SENP7
SCHEMBL9817762 0.85 MAPT (0.35) NPC1TP53GLARAB9ACYP3A4
SCHEMBL9817728 0.85 TSHR (0.37) HPGDTDP1RAB9ACYP3A4RARA
SCHEMBL9302667 0.83 KMT2A (0.40) HPGDNPC1TP53GLARAB9A
SCHEMBL9303247 0.80 CYP3A4 (0.35) HPGDNPC1TP53GLARAB9A
SCHEMBL9817687 0.80 FFAR1 (0.37) NPC1TP53GLARAB9AFFAR1
SCHEMBL8565252 0.80 KMT2A (0.45) HPGDNPC1TP53GLARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed