SCHEMBL9817635

SCHEMBL9817635

CCOC(=O)CCCCc1ccccc1C#Cc1ccc2c(c1)C(SC)(SC)CCO2

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 2/20 0.41
CYP4A11 Q02928 2/20 0.41
FAAH O00519 1/20 0.35
MGLL Q99685 1/20 0.35
FFAR1 O14842 6/20 0.34
PTGER4 P35408 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
S1PR5 Q9H228 2/20 0.33
DRD2 P14416 1/20 0.32
FFAR4 Q5NUL3 2/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817696 0.97 CYP4F2 (0.38) CYP4F2CYP4A11FFAR1PTGER4CYP1A2
SCHEMBL9817771 0.94 CYP4F2 (0.39) CYP4F2CYP4A11FFAR1S1PR5FFAR4
SCHEMBL9817669 0.89 CYP4F2 (0.43) CYP4F2CYP4A11FAAHMGLLFFAR1
SCHEMBL9817664 0.89 HPGD (0.35) FFAR1CYP3A4S1PR5
SCHEMBL9817856 0.87 CYP4Z1 (0.38) CYP4F2CYP4A11FAAHMGLLFFAR1
SCHEMBL9817777 0.86 PPARA (0.35) CYP4F2CYP4A11FAAHMGLLFFAR1
SCHEMBL9817603 0.86 CYP4F2 (0.40) CYP4F2CYP4A11FFAR1PTGER4CYP1A2
SCHEMBL9817683 0.84 CYP4Z1 (0.37) CYP4F2CYP4A11FAAHMGLLFFAR1
SCHEMBL6665905 0.84 CYP3A4 (0.37) CYP4F2CYP4A11PTGER4CYP3A4SMN1; SMN2
SCHEMBL9817649 0.84 ALOX5 (0.36) CYP4F2CYP4A11FFAR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed