SCHEMBL9817786

SCHEMBL9817786

CC(=O)OCc1ccc(C#Cc2ccc3c(c2)C(C)(C)CCO3)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.45
CYP26B1 Q9NR63 1/20 0.45
CYP3A4 P08684 3/20 0.45
RARB P10826 9/20 0.43
RARG P13631 9/20 0.43
RARA P10276 8/20 0.43
ACACB O00763 5/20 0.43
CRABP2 P29373 1/20 0.43
RXRA P19793 2/20 0.41
HNF4A P41235 1/20 0.39
SSTR5 P35346 2/20 0.38
ALDH1A1 P00352 1/20 0.38
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665705 0.88 RARA (0.49) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL9485574 0.84 RARB (0.60) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL9817629 0.83 CYP26A1 (0.45) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL9817847 0.82 CYP4F2 (0.43) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL8559730 0.81 RARB (0.54) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL9817748 0.80 CYP26A1 (0.41) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL6037049 0.80 RARB (0.67) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL9817759 0.79 CYP26A1 (0.40) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL9139588 0.79 RARA (0.44) CYP26A1CYP26B1CYP3A4RARBRARG
SCHEMBL10693553 0.78 RARB (0.73) CYP26A1CYP26B1CYP3A4RARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed