SCHEMBL9817847

SCHEMBL9817847

CCOC(=O)CCc1ccc(C#Cc2ccc3c(c2)C(C)(C)CCO3)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
CYP26A1 O43174 2/20 0.42
CYP26B1 Q9NR63 1/20 0.42
RARA P10276 5/20 0.40
RARB P10826 5/20 0.40
RARG P13631 5/20 0.40
CYP3A4 P08684 2/20 0.40
KMT2A Q03164 1/20 0.40
RXRA P19793 1/20 0.40
HNF4A P41235 1/20 0.40
CRABP2 P29373 1/20 0.39
FFAR1 O14842 5/20 0.38
ACACB O00763 2/20 0.38
CYP4Z1 Q86W10 1/20 0.37
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817748 0.94 CYP26A1 (0.41) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL9817759 0.93 CYP26A1 (0.40) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL10568461 0.91 RARA (0.39) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL9817653 0.85 CYP4F2 (0.41) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL9817640 0.85 ALOX5 (0.38) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL9817779 0.85 RARA (0.37) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL9180384 0.84 CYP4F2 (0.43) CYP4F2CYP4A11CYP26A1RARARARB
SCHEMBL8559730 0.83 RARB (0.54) CYP26A1CYP26B1RARARARBRARG
SCHEMBL6669581 0.83 RARA (0.49) CYP4F2CYP4A11CYP26A1CYP26B1RARA
SCHEMBL9817608 0.83 RARA (0.42) CYP26A1CYP26B1RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed