SCHEMBL9817812

SCHEMBL9817812

CC1(C)CCOc2ccc(C#Cc3ccc(C=O)cc3)cc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RARB P10826 11/20 0.48
RARG P13631 11/20 0.48
RARA P10276 8/20 0.48
CYP26A1 O43174 2/20 0.42
CYP3A4 P08684 1/20 0.42
CRABP2 P29373 1/20 0.42
RXRA P19793 2/20 0.40
CYP26B1 Q9NR63 1/20 0.38
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GRM5 P41594 1/20 0.34
ACACB O00763 2/20 0.33
AKR1B1 P15121 1/20 0.33
HNF4A P41235 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6665791 0.86 RARB (0.46) RARBRARGRARACYP26A1CYP3A4
SCHEMBL289444 0.84 RARB (0.55) RARBRARGRARACYP26A1RXRA
SCHEMBL6037049 0.81 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9484730 0.80 RARB (0.62) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9817629 0.79 CYP26A1 (0.45) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9817831 0.78 RARB (0.40) RARBRARGRARACYP26A1CYP3A4
SCHEMBL3521982 0.76 ALDH1A1 (0.47) RARBRARGRARACYP26A1RXRA
SCHEMBL10693990 0.76 RARB (0.80) RARBRARGRARACYP26A1CYP3A4
SCHEMBL10693994 0.76 RARB (0.80) RARBRARGRARACYP26A1CYP3A4
SCHEMBL9817786 0.76 CYP26A1 (0.45) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed