SCHEMBL9817836

SCHEMBL9817836

CCOC(=O)c1ccc(C#Cc2cc3c(cc2CC)SCCC3(C)C)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 14/20 0.61
RARA P10276 13/20 0.61
RARG P13631 11/20 0.61
CYP3A4 P08684 3/20 0.61
KMT2A Q03164 1/20 0.61
CYP26A1 O43174 2/20 0.46
CRABP2 P29373 1/20 0.40
RXRA P19793 2/20 0.39
PRKCG P05129 1/20 0.37
PRKCB P05771 1/20 0.37
PRKCA P17252 1/20 0.37
PRKCE Q02156 1/20 0.37
PRKCD Q05655 1/20 0.37
MMP13 P45452 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ESR1 P03372 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817808 0.93 RARB (0.58) RARBRARARARGCYP3A4KMT2A
SCHEMBL9817784 0.92 RARB (0.61) RARBRARARARGCYP3A4KMT2A
SCHEMBL7655154 0.90 RARA (0.50) RARBRARARARGCYP3A4KMT2A
SCHEMBL9817738 0.90 RARB (0.55) RARBRARARARGCYP3A4KMT2A
SCHEMBL444860 0.87 RARB (0.78) RARBRARARARGCYP3A4KMT2A
SCHEMBL9007003 0.87 RARB (0.66) RARBRARARARGCYP3A4KMT2A
SCHEMBL9817660 0.87 RARA (0.49) RARBRARARARGCYP3A4KMT2A
SCHEMBL6689597 0.85 RARA (0.75) RARBRARARARGCYP3A4KMT2A
SCHEMBL9180592 0.84 RARA (0.46) RARBRARARARGCYP3A4KMT2A
SCHEMBL9817823 0.84 RARB (0.47) RARBRARARARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed