SCHEMBL9817871

SCHEMBL9817871

CCOC(=O)c1cccc(C#Cc2ccc3c(c2)C(C)(C)CCS3)c1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RARA P10276 11/20 0.71
RARB P10826 11/20 0.71
RARG P13631 9/20 0.71
CYP3A4 P08684 3/20 0.71
KMT2A Q03164 1/20 0.71
CYP26A1 O43174 2/20 0.54
ACACB O00763 1/20 0.48
RXRA P19793 2/20 0.41
CRABP2 P29373 1/20 0.40
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL444860 0.90 RARB (0.78) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817655 0.88 RARA (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342992 0.86 RARA (0.69) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342924 0.85 RARB (0.68) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342993 0.85 RARA (0.68) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817758 0.85 RARA (0.62) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342899 0.85 RARB (0.79) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342915 0.83 RARB (0.66) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342967 0.83 RARB (0.66) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817722 0.83 RARA (0.63) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed