SCHEMBL9817907

SCHEMBL9817907

CCOC(=O)c1ccccc1C#Cc1cc2c(cc1SC)OCCC2(SC)SC

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
TSHR P16473 4/20 0.38
LMNA P02545 3/20 0.38
NPSR1 Q6W5P4 2/20 0.38
L3MBTL1 Q9Y468 5/20 0.34
MAPT P10636 4/20 0.34
KDM4E B2RXH2 3/20 0.34
TDP1 Q9NUW8 1/20 0.34
THRB P10828 1/20 0.34
HSD17B10 Q99714 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GAA P10253 1/20 0.32
RXRA P19793 1/20 0.32
HNF4A P41235 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
HPGD P15428 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817728 0.86 TSHR (0.37) ALDH1A1TSHRLMNANPSR1L3MBTL1
SCHEMBL9817790 0.85 MAPT (0.38) ALDH1A1TSHRLMNANPSR1L3MBTL1
SCHEMBL9817661 0.85 ACACB (0.39) ALDH1A1LMNAMAPTKDM4EMAPK1
SCHEMBL1485835 0.82 KMT2A (0.47) ALDH1A1TSHRLMNAMAPTKDM4E
SCHEMBL9817718 0.80 FDFT1 (0.38) ALDH1A1TSHRLMNANPSR1MAPT
SCHEMBL9817878 0.78 RXRA (0.44) ALDH1A1TSHRLMNANPSR1L3MBTL1
SCHEMBL9817834 0.77 ACACB (0.31)
SCHEMBL9304106 0.77 NPC1 (0.33) ALDH1A1NPSR1L3MBTL1MAPTSMN1; SMN2
SCHEMBL6665869 0.75 CYP4F2 (0.30)
SCHEMBL6667812 0.75 CYP4F2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed