SCHEMBL9817878

SCHEMBL9817878

CCOC(=O)c1ccccc1C#Cc1cc2c(cc1C)OCCC2(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.44
HNF4A P41235 1/20 0.44
TSHR P16473 3/20 0.40
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
THRB P10828 1/20 0.38
RARA P10276 6/20 0.37
RARB P10826 6/20 0.37
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
RARG P13631 5/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CYP3A4 P08684 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP26A1 O43174 1/20 0.34
CYP26B1 Q9NR63 1/20 0.34
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817712 0.87 RARA (0.44) RXRAHNF4ATSHRLMNAMAPT
SCHEMBL10571276 0.84 RARA (0.46) RXRAHNF4ATSHRLMNAMAPT
SCHEMBL9817818 0.83 RARA (0.42) RXRAHNF4ALMNAMAPTRARA
SCHEMBL9142284 0.82 RXRA (0.41) RXRAHNF4ALMNAMAPTRARA
SCHEMBL9138172 0.82 RXRA (0.41) RXRAHNF4ALMNAMAPTRARA
SCHEMBL6668066 0.81 RARA (0.57) RXRAHNF4ATSHRLMNAMAPT
SCHEMBL9817900 0.80 RARA (0.47) RXRATSHRLMNAMAPTRARA
SCHEMBL9817887 0.78 RXRA (0.41) RXRAHNF4AMAPTRARARARB
SCHEMBL9817907 0.78 ALDH1A1 (0.38) RXRAHNF4ATSHRLMNAMAPT
SCHEMBL9137414 0.77 RXRA (0.39) RXRAHNF4AMAPTRARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed