SCHEMBL9822989

SCHEMBL9822989

O=C(NC(CC1=CCCCC1)C1CCCN1)c1cc(Cl)cc2c1OCC2

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.42
CXCR3 P49682 1/20 0.32
MAPT P10636 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NFKB1 P19838 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9822819 0.96 HTR3A (0.37) HTR3ACXCR3MAPTNPC1ALDH1A1
Fumaric Acid SCHEMBL9868273 0.91 HTR3A (0.35) HTR3A
SCHEMBL9822707 0.86 TP53 (0.33) CXCR3
Hydrochloric Acid SCHEMBL9406910 0.84 HTR3A (0.45) HTR3A
SCHEMBL9822695 0.82 SMN1; SMN2 (0.32) ALDH1A1
SCHEMBL9822842 0.82 ALDH1A1 (0.31) MAPTALDH1A1
SCHEMBL10369470 0.77 SMN1; SMN2 (0.32) ALDH1A1
SCHEMBL10424728 0.75 BACE1 (0.34) HTR3A
Hydrochloric Acid SCHEMBL7264982 0.74 BACE1 (0.34) HTR3A
SCHEMBL7272680 0.74 PARP1 (0.33) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0231139-B1 DIHYDROBENZOFURANE AND CHROMANE CARBOXAMIDE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS NEUROLEPTICS Laboratoires DELAGRANGE (FR) 1991-12-04 EP claimed
US-5006570-A Dihydrobenzofuran- and chroman-carboxamide derivatives, processes for the preparation thereof and use thereof as neuroleptics LABORATOIRES DELAGRANGE (FR) 1991-04-09 US disclosed