SCHEMBL9823028

SCHEMBL9823028

CC(=O)c1ccc2nc3c(nc2c1)CCCC3

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.51
NPC1 O15118 5/20 0.48
RAB9A P51151 4/20 0.48
HPGD P15428 2/20 0.47
MAPT P10636 4/20 0.47
POLB P06746 2/20 0.47
BLM P54132 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
BCHE P06276 3/20 0.46
ACHE P22303 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 4/20 0.43
GRM1 Q13255 2/20 0.42
APP P05067 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565647 0.84 TDP1 (0.61) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL9822779 0.78 TDP1 (0.72) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL9091793 0.77 TDP1 (0.50) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL24931057 0.76 MAPT (0.77) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL9748752 0.76 ACHE (0.72) BCHEACHE
SCHEMBL9822932 0.74 CYP2A6 (0.49) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL9823025 0.74 NPC1 (0.75) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL30134026 0.72 TDP1 (0.46) KMT2ANPC1RAB9AHPGDMAPT
SCHEMBL22237575 0.72 TDP1 (0.46) NPC1RAB9AHPGDMAPTTDP1
SCHEMBL24920215 0.72 NPC1 (0.54) KMT2ANPC1RAB9AHPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288898-B1 SUBSTITUTED CHINOXALYL-IMIDAZOLIDINE-2,4-DIONES, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND PHARMACOLOGICAL PREPARATIONS HOECHST AKTIENGESELLSCHAFT (DE) 1991-08-14 EP disclosed
US-4943576-A ENZYME INHIBITORS HOECHST AKTIENGESELLSCHAFT (DE) 1990-07-24 US disclosed
EP-0288898-A1 Substituted chinoxalyl-imidazolidine-2,4-diones, process for their preparation, their use as medicaments and pharmacological preparations HOECHST AKTIENGESELLSCHAFT (DE) 1988-11-02 EP disclosed