SCHEMBL9823481

SCHEMBL9823481

Nc1nc2ccc(CNCC#Cc3ccc(Cl)c(Cl)c3)cc2c(=O)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TYMS P04818 3/20 0.43
DHFR P00374 7/20 0.43
ATIC P31939 1/20 0.40
PNP P00491 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823104 0.86 DHFR (0.44) TYMSDHFRATIC
SCHEMBL9823281 0.83 DHFR (0.56) TYMSDHFRATIC
SCHEMBL9823454 0.82 DHFR (0.55) TYMSDHFRATIC
SCHEMBL9823232 0.82 MEN1 (0.36) TYMS
SCHEMBL9823450 0.82 IP6K1 (0.47) DHFR
SCHEMBL9823195 0.81 DHFR (0.45) TYMSDHFRATIC
SCHEMBL9823278 0.79 DHFR (0.47) TYMSDHFR
SCHEMBL9823478 0.77 DHFR (0.44) TYMSDHFR
SCHEMBL9823634 0.76 DHFR (0.43) TYMSDHFR
SCHEMBL28787846 0.74 TYMS (0.54) TYMSDHFRATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP claimed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US claimed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP claimed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO claimed
EP-0426666-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1991-05-15 EP disclosed
US-4857530-A THYMIDYLATE SYNTHASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1989-08-15 US disclosed
EP-0316657-A1 Substituted quinazolinones as anticancer agents WARNER-LAMBERT COMPANY (US) 1989-05-24 EP disclosed
WO-1989004307-A1 SUBSTITUTED QUINAZOLINONES AS ANTICANCER AGENTS WARNER-LAMBERT COMPANY (US) 1989-05-18 WO disclosed