SCHEMBL9824026

SCHEMBL9824026

CC(C)(Cc1ccc(OC(F)(F)F)cc1)C(=O)Cn1cncn1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
CYP19A1 P11511 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
ABL1 P00519 3/20 0.40
BCR P11274 3/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
EPHX2 P34913 1/20 0.39
NR1H4 Q96RI1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9272650 0.85 CYP3A4 (0.43) CYP1A2CYP3A4CYP2D6CYP2C19PPARD
SCHEMBL9022060 0.83 CYP3A4 (0.45) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL9871573 0.83 CYP3A4 (0.52) CYP1A2CYP3A4CYP2D6CYP2C19CYP19A1
SCHEMBL9823992 0.82 KDM4A (0.38) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL9203686 0.82 CYP3A4 (0.41) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL10726056 0.82 CYP19A1 (0.50) CYP1A2CYP3A4CYP2D6CYP2C19CYP19A1
SCHEMBL10333953 0.81 LMNA (0.40) CYP1A2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL9824107 0.80 TSHR (0.46) CYP1A2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL9823573 0.77 CYP19A1 (0.53) CYP1A2CYP3A4CYP2D6CYP2C19CYP2C9
SCHEMBL3319305 0.75 CYP19A1 (0.57) CYP1A2CYP3A4CYP2D6CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301393-B1 1,4-DISUBSTITUTED 1-AZOLYL-3,3-DYMETHYLBUTANE DERIVATIVES BAYER AG (DE) 1991-08-14 EP disclosed
US-4968712-A PHYTOPATHOGENS, AGRICULTURE BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed
EP-0301393-A1 1,4-Disubstituted 1-azolyl-3,3-dymethylbutane derivatives BAYER AG (DE) 1989-02-01 EP disclosed