SCHEMBL9823573

SCHEMBL9823573

O=C(Cn1cncn1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.53
CYP11B1 P15538 2/20 0.53
CYP11B2 P19099 2/20 0.53
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
LMNA P02545 1/20 0.46
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10559569 0.83 ALDH1A1 (0.55) MAPTHTTLMNAHDAC1HDAC6
SCHEMBL9864864 0.83 PTPN1 (0.49) CYP19A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL673406 0.81 LMNA (0.53) CYP19A1CYP11B1CYP11B2CYP3A4CYP2C9
SCHEMBL17208333 0.81 KDM4E (0.50) CYP19A1CYP11B1CYP11B2MAPTHTT
SCHEMBL16563433 0.80 CYP19A1 (0.52) CYP19A1CYP11B1CYP11B2HTR2AHTR2C
SCHEMBL8137901 0.78 L3MBTL1 (0.54) CYP19A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13781424 0.78 HDAC1 (0.50) CYP19A1CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7293623 0.78 HTT (0.63) CYP19A1MAPTHTTLMNAHDAC1
SCHEMBL412906 0.78 HDAC1 (0.49) CYP19A1MAPTHTTHDAC1HDAC6
SCHEMBL6558375 0.78 CYP1A2 (0.59) CYP19A1CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0174769-B1 ANTIFUNGAL AZOLE COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-11-21 EP disclosed
US-4925863-A 1,3-DI(1,2,4-TRIAZOL-1-YL)-2-PROPANOL DERIVATIVES SUBSTITUTED WITH A STYRYL GROUP IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-05-15 US disclosed
EP-0174769-A1 Antifungal azole compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-03-19 EP disclosed