SCHEMBL9824575

SCHEMBL9824575

CCn1c2s[nH]c(=O)c2c(=O)c2cc(F)c(N3CCC(N)C3)c(Cl)c21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
PIM1 P11309 2/20 0.42
GSK3A P49840 2/20 0.42
GSK3B P49841 1/20 0.42
PIM3 Q86V86 1/20 0.42
CSNK1G1 Q9HCP0 1/20 0.42
TOP1 P11387 2/20 0.40
IKBKB O14920 1/20 0.40
AURKA O14965 1/20 0.40
CHUK O15111 1/20 0.40
MAPK13 O15264 1/20 0.40
DAPK3 O43293 1/20 0.40
PRKCG P05129 1/20 0.40
CDK2 P24941 1/20 0.40
MARK3 P27448 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209335 0.93 PIM1 (0.47) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824957 0.86 ALDH1A1 (0.54) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824350 0.85 KDM4E (0.49) ALDH1A1POLBOPRM1PIM1GSK3A
SCHEMBL9824362 0.84 PIM1 (0.37) ALDH1A1PIM1GSK3APIM3IKBKB
SCHEMBL9824172 0.84 KDM4E (0.40) ALDH1A1PIM1GSK3APIM3IKBKB
SCHEMBL9824748 0.84 ALDH1A1 (0.49) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824259 0.83 ALDH1A1 (0.47) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9214069 0.82 KCNH2 (0.44) ALDH1A1PIM1GSK3ATOP1IKBKB
SCHEMBL9824093 0.81 PRKD3 (0.47) PIM1GSK3AGSK3BPIM3TOP1
SCHEMBL9215159 0.80 PIM1 (0.56) PIM1GSK3AGSK3BPIM3CSNK1G1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed