SCHEMBL9824259

SCHEMBL9824259

NC1CCN(c2c(F)cc3c(=O)c4c(=O)[nH]sc4n(-c4ccc(F)cc4)c3c2Cl)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
CHRM2 P08172 1/20 0.47
CHRM1 P11229 1/20 0.47
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
TOP1 P11387 2/20 0.40
PIM1 P11309 2/20 0.38
GSK3A P49840 2/20 0.38
IKBKB O14920 1/20 0.38
AURKA O14965 1/20 0.38
CHUK O15111 1/20 0.38
MAPK13 O15264 1/20 0.38
DAPK3 O43293 1/20 0.38
PRKCG P05129 1/20 0.38
CDK2 P24941 1/20 0.38
MARK3 P27448 1/20 0.38
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
MAPKAPK2 P49137 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824479 0.85 KDM4E (0.36) ALDH1A1PIM1GSK3AIKBKBAURKA
SCHEMBL9824962 0.84 ALK (0.39) ALDH1A1PIM1GSK3AIKBKBAURKA
SCHEMBL9824957 0.84 ALDH1A1 (0.54) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824885 0.83 ALDH1A1 (0.48) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824575 0.83 ALDH1A1 (0.49) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9824308 0.81 PRKD3 (0.43) TOP1PIM1GSK3AGSK3BPIM3
SCHEMBL9823968 0.80 KMT2A (0.49)
SCHEMBL9839117 0.78 TOP2A (0.40) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL9209335 0.78 PIM1 (0.47) ALDH1A1POLBCHRM2CHRM1OPRM1
Hydrochloric Acid SCHEMBL9839687 0.77 TOP2A (0.39) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed