SCHEMBL9824618

SCHEMBL9824618

CCN(CC)CCC1CCCCN1CC(=O)NC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
S1PR1 P21453 3/20 0.37
S1PR3 Q99500 3/20 0.37
S1PR5 Q9H228 3/20 0.37
TSHR P16473 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 3/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 2/20 0.33
ALOX15 P16050 2/20 0.33
S1PR4 O95977 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
MAPK1 P28482 1/20 0.32
TERT O14746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824251 0.86 CYP1A2 (0.41) ALDH1A1TSHRNPSR1KMT2APOLB
SCHEMBL9824048 0.83 S1PR1 (0.36) ALDH1A1S1PR1S1PR3S1PR5TSHR
SCHEMBL18878632 0.81 LTA4H (0.39) ALDH1A1TSHRNPSR1KMT2APOLB
SCHEMBL9245124 0.80 ALDH1A1 (0.38) ALDH1A1S1PR1S1PR3S1PR5TSHR
SCHEMBL28296702 0.79 ALDH1A1 (0.37) ALDH1A1S1PR1S1PR3S1PR5TSHR
SCHEMBL9824064 0.77 LTA4H (0.40) ALDH1A1TSHRNPSR1KMT2APOLB
SCHEMBL9824639 0.76 S1PR1 (0.42) ALDH1A1S1PR1S1PR3S1PR5TSHR
SCHEMBL9824284 0.76 S1PR1 (0.40) ALDH1A1S1PR1S1PR3S1PR5TSHR
SCHEMBL27799980 0.74 ALDH1A1 (0.41) ALDH1A1S1PR1S1PR3S1PR5TSHR
SCHEMBL9824423 0.73 S1PR1 (0.38) S1PR1S1PR3S1PR5S1PR4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273239-B1 CONDENSED DIAZEPINONES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1991-03-06 EP disclosed
US-4873236-A BRADYCARDIAL AGENTS DR. KARL THOMAE GMBH (DE) 1989-10-10 US disclosed
EP-0273239-A1 Condensed diazepinones, processes for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1988-07-06 EP disclosed