SCHEMBL9824874

SCHEMBL9824874

O=c1[nH]oc2c1c(=O)c1cc(F)c(N3CCNCC3)c(Cl)c1n2C1CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
POLB P06746 2/20 0.38
OPRM1 P35372 2/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
OPRD1 P41143 1/20 0.38
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 3/20 0.38
KCNH2 Q12809 2/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2D6 P10635 1/20 0.38
CACNA1C Q13936 1/20 0.38
SCN5A Q14524 1/20 0.38
TOP2A P11388 5/20 0.35
TOP2B Q02880 4/20 0.35
HSD17B10 Q99714 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
LMNA P02545 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824684 0.90 TOP2A (0.36) ALDH1A1POLBOPRM1CYP1A2CYP2C9
SCHEMBL9824167 0.89 CYP1A2 (0.39) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9824506 0.88 ALDH1A1 (0.38) ALDH1A1POLBOPRM1CYP1A2CYP2C9
SCHEMBL9823991 0.88 ALDH1A1 (0.46) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9824606 0.85 ALDH1A1 (0.55) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9824851 0.82 PIM1 (0.40) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9824776 0.82 ALDH1A1 (0.40) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9825005 0.81 IKBKB (0.50) IKBKBAURKACHUKMAPK13DAPK3
SCHEMBL9824887 0.80 ALDH1A1 (0.36) ALDH1A1POLBOPRM1CHRM2CHRM1
SCHEMBL9825033 0.80 KDM4E (0.43) ALDH1A1POLBTOP2AHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed