SCHEMBL9824915

SCHEMBL9824915

CC1CN(c2nc3c(cc2F)c(=O)c2c(=O)[nH]oc2n3-c2ccc(F)cc2)CCN1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HPGD P15428 4/20 0.35
KDM4E B2RXH2 3/20 0.35
HSD17B10 Q99714 3/20 0.35
KMT2A Q03164 2/20 0.34
LMNA P02545 2/20 0.34
CYP2C9 P11712 1/20 0.34
ATP6V1B2 P21281 1/20 0.34
TBXA2R P21731 1/20 0.34
EDNRA P25101 1/20 0.34
TARBP2 Q15633 1/20 0.34
PMP22 Q01453 1/20 0.34
BCL2A1 Q16548 2/20 0.33
KHK P50053 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
PRKD3 O94806 1/20 0.33
ALOX15 P16050 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824747 0.85 KMT2A (0.49) ALDH1A1HPGDKDM4EHSD17B10KMT2A
SCHEMBL9824797 0.85 TNKS (0.39) KMT2ALMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL9824035 0.83 KDM4E (0.39) ALDH1A1HPGDKDM4EHSD17B10KMT2A
SCHEMBL9824254 0.83 KMT2A (0.34) KMT2ALMNACYP2C9ATP6V1B2TBXA2R
SCHEMBL9823980 0.82 KDM4E (0.42) ALDH1A1HPGDKDM4EHSD17B10KMT2A
SCHEMBL9824600 0.76 KCNH2 (0.36) ALDH1A1HPGDKDM4EHSD17B10KMT2A
Hydrochloric Acid SCHEMBL10766907 0.75 KMT2A (0.58) ALDH1A1HPGDKDM4EHSD17B10KMT2A
SCHEMBL10669165 0.75 EPHA2 (0.45) ALDH1A1HPGDKDM4EHSD17B10KMT2A
SCHEMBL10577440 0.73 PDE7A (0.34) HPGD
SCHEMBL9824114 0.73 ALDH1A1 (0.41) ALDH1A1HPGDKDM4EHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed