SCHEMBL9824747

SCHEMBL9824747

NC1CCN(c2nc3c(cc2F)c(=O)c2c(=O)[nH]oc2n3-c2ccc(F)cc2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.49
HRH4 Q9H3N8 2/20 0.40
DPP4 P27487 2/20 0.37
EPHA2 P29317 1/20 0.36
FLT4 P35916 1/20 0.36
GSK3B P49841 1/20 0.36
RARB P10826 1/20 0.36
TBXAS1 P24557 1/20 0.36
SLC6A3 Q01959 1/20 0.36
MAT2A P31153 1/20 0.36
RPS6KB1 P23443 1/20 0.34
MATK P42679 1/20 0.34
DYRK1A Q13627 1/20 0.34
MAPKAPK3 Q16644 1/20 0.34
PIM3 Q86V86 1/20 0.34
AURKB Q96GD4 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10766907 0.90 KMT2A (0.58) KMT2AHRH4DPP4EPHA2FLT4
SCHEMBL9824915 0.85 ALDH1A1 (0.35) KMT2ADPP4EPHA2FLT4GSK3B
SCHEMBL9824797 0.84 TNKS (0.39) KMT2AHRH4LMNA
SCHEMBL9824074 0.84 KMT2A (0.46) KMT2AHRH4DPP4GSK3BMAT2A
SCHEMBL9823968 0.82 KMT2A (0.49) KMT2AHRH4DPP4
SCHEMBL9824004 0.82 TOP1 (0.43) KMT2AGSK3BDYRK1APIM3KDM4E
SCHEMBL9825021 0.82 PIM1 (0.43) GSK3BPIM3ALDH1A1POLBTOP2A
SCHEMBL9824535 0.82 KMT2A (0.45) KMT2AHRH4DPP4GSK3BMAT2A
SCHEMBL10577440 0.81 PDE7A (0.34) HPGD
SCHEMBL9824885 0.81 ALDH1A1 (0.48) GSK3BPIM3ALDH1A1POLBTOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0227088-B1 ISOXAZOLO-NAPHTHYRIDINE, ISOXAZOLO QUINOLINE, ISOTHIAZOLONAPHTHYRIDINE, AND ISOTHIAZOLOQUINOLINE DERIVATIVES ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
US-4767762-A Tricyclic quinoline and naphthyride antibacterials ABBOTT LABORATORIES (US) 1988-08-30 US disclosed
EP-0227088-A1 Isoxazolo-naphthyridine, isoxazolo quinoline, isothiazolonaphthyridine, and isothiazoloquinoline derivatives ABBOTT LABORATORIES (US) 1987-07-01 EP disclosed