SCHEMBL9825409

SCHEMBL9825409

ClCCCOc1ccc2c(c1)OCC=C2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 1/20 0.54
MAOB P27338 12/20 0.40
MAOA P21397 6/20 0.38
TSHR P16473 2/20 0.35
CA12 O43570 1/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
PPARG P37231 3/20 0.32
PPARD Q03181 3/20 0.32
FFAR1 O14842 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21365816 0.84 STS (0.50) STSTSHR
SCHEMBL14515202 0.81 STS (0.53) STSMAOBMAOATSHRCA12
SCHEMBL27397632 0.79 STS (0.60) STS
SCHEMBL22916225 0.78 CA12 (0.56) STSMAOBMAOATSHRCA12
SCHEMBL11010282 0.77 MAOB (0.58) STSMAOBMAOACA12CA9
SCHEMBL28445528 0.76 STS (0.60) STSCA12CA9MEN1CYP3A4
SCHEMBL29634256 0.76 STS (0.60) STSCA12CA9MEN1CYP3A4
SCHEMBL7236239 0.72 MAOB (0.71) MAOBMAOATSHRMEN1CYP1A2
SCHEMBL27353149 0.71 STS (0.55) STSTSHRMEN1MAPTKMT2A
SCHEMBL30421522 0.70 STS (0.53) STSMEN1MAPTMAPK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237781-B1 PHENYL AND HETEROCYCLIC TETRAHYDROPYRIDYL AND PIPERAZINYL ALKOXY-BENZHETEROCYCLIC COMPOUNDS AS ANTIPSYCHOTIC AGENTS WARNER-LAMBERT COMPANY (US) 1991-04-24 EP disclosed
US-4803203-A SCHIZOPHRENIA, NEUOLEPTIC AGENTS WARNER-LAMBERT COMPANY (US) 1989-02-07 US disclosed
US-4704390-A SCHIZOPHRENIA WARNER-LAMBERT COMPANY (US) 1987-11-03 US disclosed
EP-0237781-A2 Phenyl and heterocyclic tetrahydropyridyl and piperazinyl alkoxy-benzheterocyclic compounds as antipsychotic agents WARNER-LAMBERT COMPANY (US) 1987-09-23 EP disclosed