SCHEMBL9825792

SCHEMBL9825792

COC(=O)c1ccc(CCN(C)CCO)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 4/20 0.64
CYP4F2 P78329 3/20 0.62
LOXL2 Q9Y4K0 1/20 0.51
THRA P10827 1/20 0.50
THRB P10828 1/20 0.50
ALDH1A1 P00352 4/20 0.49
HPGD P15428 2/20 0.49
HSD17B10 Q99714 2/20 0.49
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
GAA P10253 1/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24835147 0.86 CYP4A11 (0.57) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL5776546 0.86 CYP4A11 (0.57) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL15329199 0.83 CYP4A11 (0.62) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL24835284 0.82 CYP4A11 (0.60) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL2655571 0.81 CYP4A11 (0.79) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL9826363 0.81 SMN1; SMN2 (0.58) CYP4A11CYP4F2ALDH1A1KDM4ETSHR
SCHEMBL70185 0.79 CYP4A11 (0.75) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL2654777 0.78 CYP4A11 (1.00) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL24835214 0.78 CYP4A11 (0.58) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL5068476 0.78 CYP4A11 (0.68) CYP4A11CYP4F2LOXL2THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0239815-B1 SUBSTITUTED THIAZOLES AND OXAZOLES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1991-07-24 EP disclosed
EP-0239815-A1 Substituted thiazoles and oxazoles, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-10-07 EP disclosed