SCHEMBL9826015

SCHEMBL9826015

COC1=NOC(CNC(=O)OC(C)(C)C)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MIF P14174 2/20 0.42
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
EPHX1 P07099 1/20 0.35
LMNA P02545 1/20 0.35
GFER P55789 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
ACACB O00763 2/20 0.35
ACACA Q13085 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
CTSK P43235 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12449472 0.86 MIF (0.40) MIFHTTNPSR1MEN1KMT2A
SCHEMBL2034511 0.83 MIF (0.43) MIFHTTNPSR1EPHX1LMNA
SCHEMBL9825924 0.82 MIF (0.45) MIFHTTNPSR1GAAEPHX1
SCHEMBL4610456 0.77 MIF (0.40) MIFHTTNPSR1GAAEPHX1
SCHEMBL9825478 0.77 MIF (0.40) MIFHTTNPSR1MEN1KMT2A
SCHEMBL18669141 0.75 GAA (0.41) GAACTSK
SCHEMBL590406 0.74 HCRTR2 (0.47) HTTNPSR1MEN1GAAKMT2A
SCHEMBL590405 0.74 HCRTR2 (0.47) HTTNPSR1MEN1GAAKMT2A
SCHEMBL2750096 0.74 HCRTR2 (0.47) HTTNPSR1MEN1GAAKMT2A
SCHEMBL28662052 0.71 HCRTR2 (0.45) HTTSMN1; SMN2MEN1KMT2AEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237082-B1 3,5-DISUBSTITUTED 4,5-DIHYDROISOXAZOLES AS TRANSGLUTAMINASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1991-05-29 EP disclosed
US-4929630-A SKIN DISORDERS, ACNE, 4,5-DIHYDROISOOXAZOLE PEPTIDES SYNTEX (U.S.A.) INC. (US) 1990-05-29 US disclosed
US-4912120-A Containing amine and amide substitution SYNTEX (U.S.A.) INC. (US) 1990-03-27 US disclosed
EP-0237082-A2 3,5-disubstituted 4,5-dihydroisoxazoles as transglutaminase inhibitors SYNTEX (U.S.A.) INC. (US) 1987-09-16 EP disclosed