SCHEMBL9828090

SCHEMBL9828090

COS(=O)(=O)O.c1ccc(CNCc2ccccc2)cc1

nearest known ligand 0.53

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.53
CA1 P00915 4/20 0.53
SMN1; SMN2 Q16637 1/20 0.50
HTT P42858 1/20 0.49
CA12 O43570 2/20 0.48
CA7 P43166 2/20 0.48
CA14 Q9ULX7 2/20 0.48
MAOA P21397 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
CHRM2 P08172 1/20 0.47
ATM Q13315 1/20 0.46
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
BCHE P06276 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfuric Acid SCHEMBL9523490 0.86 CA2 (0.61) CA2CA1CA12CA7CA14
Sulfuric Acid SCHEMBL9523482 0.86 CA2 (0.61) CA2CA1CA12CA7CA14
SCHEMBL28471233 0.84 CA2 (0.56) CA2CA1SMN1; SMN2CA12CA7
SCHEMBL29102028 0.81 HTT (0.43) CA2CA1SMN1; SMN2HTTCA12
Methoxymethane SCHEMBL10589288 0.81 MEN1 (0.64) SMN1; SMN2HTTMAOAMEN1KMT2A
Benzyl Alcohol SCHEMBL29257722 0.80 TSHR (0.58) CA2CA1SMN1; SMN2HTTCA12
SCHEMBL14890478 0.80 SMN1; SMN2 (0.40) CA2CA1SMN1; SMN2HTTMEN1
Benzenemethanethiol SCHEMBL10351782 0.78 IDO1 (0.56) CA2CA1HTTCA12CA7
Benzylamine SCHEMBL12985628 0.78 LOXL2 (0.56) CA2CA1SMN1; SMN2CA12CA7
Phenylmethanesulfonic Acid SCHEMBL5078710 0.78 PRSS1 (0.49) CA2CA1SMN1; SMN2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0235628-B1 1-ARYLPYRAZOLES BAYER AG (DE) 1991-04-24 EP disclosed
EP-0232538-B1 5-ACYLAMIDO-1-ARYL PYRAZOLES BAYER AG (DE) 1990-05-23 EP disclosed
EP-0222253-B1 SUBSTITUTED 5-AMINO-1-ARYL-PYRAZOLES BAYER AG (DE) 1989-04-05 EP disclosed
US-4814001-A PLANT GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1989-03-21 US disclosed
US-4810283-A PRE- AND POSTEMERGENCE BAYER AKTIENGESELLSCHAFT (DE) 1989-03-07 US disclosed
EP-0173821-B1 SUBSTITUTED 5-AMINO-1-PHENYL PYRAZOLES BAYER AG (DE) 1989-01-18 EP disclosed
US-4772310-A 5-acylamino-pyrazole derivatives, composition containing them, and their use as herbicides and plant growth BAYER AKTIENGESELLSCHAFT (DE) 1988-09-20 US disclosed
US-4740232-A Substituted 5-amino-1-phenylpyrazoles composition containing them and herbicidal method of using them BAYER AKTIENGESELLSCHAFT (DE) 1988-04-26 US disclosed
US-4734125-A 5-acylamido-1-aryl-pyrazoles, composition containing them and herbicidal method of using them BAYER AKTIENGESELLSCHAFT (DE) 1988-03-29 US disclosed
EP-0257479-A1 Substituted 1-aryl-3-tert.-butyl pyrazoles BAYER AG (DE) 1988-03-02 EP disclosed
US-4695308-A Herbicidal substituted 5-amino-1-aryl-pyrazoles BAYER AKTIENGESELLSCHAFT (DE) 1987-09-22 US disclosed
EP-0235628-A2 1-Arylpyrazoles BAYER AG (DE) 1987-09-09 EP disclosed
EP-0232538-A2 5-Acylamido-1-aryl pyrazoles BAYER AG (DE) 1987-08-19 EP disclosed
EP-0173821-A1 Substituted 5-amino-1-phenyl pyrazoles BAYER AG (DE) 1986-03-12 EP disclosed