SCHEMBL9828162

SCHEMBL9828162

N=C(N)N(CCCc1c[nH]cn1)CCN(c1ccccc1)c1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
HDAC1 Q13547 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
HDAC9 Q9UKV0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9828346 0.99 FFAR1 (0.40) FFAR1FFAR4CYP2D6CYP2C19HDAC1
SCHEMBL9827728 0.92 FFAR1 (0.35) FFAR1FFAR4CYP2D6CYP2C19
Hydrochloric Acid SCHEMBL9827657 0.91 FFAR1 (0.34) FFAR1FFAR4CYP2D6CYP2C19
SCHEMBL9828326 0.90 HRH4 (0.33)
Hydrochloric Acid SCHEMBL9827568 0.89 GRIN2D (0.33)
SCHEMBL9828412 0.85 CHRM2 (0.46) CYP2D6CYP2C19
SCHEMBL7287544 0.84 HRH1 (0.41) CYP2C19
SCHEMBL9829110 0.84 SIGMAR1 (0.38)
Hydrochloric Acid SCHEMBL9827919 0.84 LMNA (0.47) CYP2D6CYP2C19
SCHEMBL9827932 0.82 CYP2D6 (0.50) CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0302896-B1 N-(W-SUBSTITUTED ALKYL)-N'-[(IMIDAZOLE-4-YL)ALKYL]GUANIDINE CEDONA PHARMACEUTICALS B.V. (NL) 1991-08-14 EP claimed