SCHEMBL9828636

SCHEMBL9828636

CNCCc1c[nH]c2ccc(C3=NCCN3)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.54
MPO P05164 3/20 0.54
HTR2C P28335 2/20 0.54
MEN1 O00255 1/20 0.54
CYP2D6 P10635 1/20 0.54
KMT2A Q03164 1/20 0.54
HTR1A P08908 3/20 0.52
HTR2A P28223 2/20 0.52
HTR1D P28221 2/20 0.52
HTR1B P28222 2/20 0.52
ALDH1A1 P00352 2/20 0.49
LMNA P02545 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
HTT P42858 1/20 0.49
NISCH Q9Y2I1 6/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNA7 P36544 1/20 0.45
CHRNA4 P43681 1/20 0.45
HTR5A P47898 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828643 0.84 HTR1D (0.59) MPOHTR2CCYP2D6HTR1AHTR2A
SCHEMBL9827561 0.84 HTR1A (0.54) MPOHTR2CCYP2D6KMT2AHTR1A
SCHEMBL9827688 0.77 HTR1D (0.50) MPOHTR2CCYP2D6KMT2AHTR1A
Hydrochloric Acid SCHEMBL10555707 0.76 HTR1A (0.50) MPOHTR2CCYP2D6KMT2AHTR1A
SCHEMBL7330504 0.76 KDM4E (0.66) KDM4EMPOHTR2CMEN1CYP2D6
SCHEMBL1935161 0.74 NISCH (0.69) HTR1DLMNANISCH
Hydrochloric Acid SCHEMBL2239536 0.72 NISCH (0.68) HTR1DLMNANISCH
Hydrochloric Acid SCHEMBL15514269 0.72 NISCH (0.68) HTR1DLMNANISCH
Hydrochloric Acid SCHEMBL1935805 0.72 NISCH (0.68) HTR1DLMNANISCH
SCHEMBL4303662 0.72 KDM4E (0.70) KDM4EMPOHTR2CMEN1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0225726-B1 INDOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1991-04-17 EP disclosed
US-4833153-A VASOCONSTRICTORS, MIGRAINES GLAXO GROUP LIMITED (GB) 1989-05-23 US disclosed
EP-0225726-A1 Indole derivatives GLAXO GROUP LIMITED (GB) 1987-06-16 EP disclosed