SCHEMBL9829147

SCHEMBL9829147

COc1ccc(OCCCN(C)CCc2ccc(OC)c(OC)c2)c(C2(SC)Sc3ccccc3N(C)C2=O)c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 9/20 0.51
ABCB1 P08183 2/20 0.44
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9832211 0.99 SMPD1 (0.50) SMPD1ABCB1CYP3A4
Hydrochloric Acid SCHEMBL9831196 0.97 SMPD1 (0.49) SMPD1ABCB1CYP3A4
SCHEMBL9828526 0.91 SMPD1 (0.42) SMPD1ABCB1
Hydrochloric Acid SCHEMBL9829234 0.90 SMPD1 (0.41) SMPD1ABCB1
Hydrochloric Acid SCHEMBL9831407 0.88 SMPD1 (0.51) SMPD1ABCB1CYP3A4
SCHEMBL9829599 0.87 SMPD1 (0.51) SMPD1ABCB1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9830009 0.86 SMPD1 (0.51) SMPD1ABCB1CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9828653 0.86 BCHE (0.36) SMPD1CYP3A4
Hydrochloric Acid SCHEMBL9828610 0.86 SMPD1 (0.46) SMPD1ABCB1CYP3A4
Hydrochloric Acid SCHEMBL9829155 0.85 SMPD1 (0.50) SMPD1ABCB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233291-B1 2-ARYLBENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1991-03-13 EP claimed
US-4739050-A CALCIUM ANTAGONIST, ANTICOAGULANT SANTEN PHARMACEUTICAL CO., LTD. (JP) 1988-04-19 US claimed
EP-0233291-A1 2-ARYLBENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1987-08-26 EP claimed
EP-0236618-A2 Insecticidal N'-substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1987-09-16 EP disclosed