SCHEMBL9829316

SCHEMBL9829316

COCCOc1cc(Cc2cnc(N)nc2N)cc2c1NCCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.52
MEN1 O00255 1/20 0.50
SLC22A1 O15245 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP3A4 P08684 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
CYP2C19 P33261 1/20 0.50
BLM P54132 1/20 0.50
KMT2A Q03164 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830401 0.90 DHFR (0.60) DHFRMEN1SLC22A1ALDH1A1CYP3A4
Tetroxoprim SCHEMBL155211 0.75 MEN1 (0.78) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL9829650 0.73 DHFR (0.54) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL9830078 0.73 DHFR (0.51) DHFR
SCHEMBL10488971 0.73 DHFR (0.81) DHFR
Hydrochloric Acid SCHEMBL9830813 0.72 DHFR (0.50) DHFR
SCHEMBL9161460 0.72 MEN1 (0.73) DHFRMEN1SLC22A1ALDH1A1CYP3A4
Aditeren SCHEMBL1230789 0.71 DHFR (0.81) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL6555239 0.71 DHFR (0.51) DHFR
Aditeren SCHEMBL10676774 0.70 DHFR (0.79) DHFRMEN1SLC22A1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US claimed
EP-0096214-B1 ANTIBACTERIAL PYRIMIDINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-02-27 EP disclosed
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US disclosed
EP-0096214-A1 Antibacterial pyrimidine compounds THE WELLCOME FOUNDATION LIMITED (GB) 1983-12-21 EP disclosed