SCHEMBL9829342

SCHEMBL9829342

Cn1nc(-c2cccnc2)nc1-c1ccccc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.48
HSD11B1 P28845 8/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46
S1PR1 P21453 1/20 0.44
TRPA1 O75762 1/20 0.43
HTT P42858 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
KCNT1 Q5JUK3 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
AHR P35869 1/20 0.42
USP1 O94782 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829470 0.86 HSD11B1 (0.50) HSD11B1NPC1RAB9ANR1H2NR1H3
SCHEMBL9830541 0.82 HSD11B1 (0.58) HSD11B1NPC1RAB9ANR1H2NR1H3
SCHEMBL9830876 0.81 HSD11B1 (0.51) HSD11B1TRPA1
SCHEMBL11589724 0.79 NR1H2 (0.61) NPC1RAB9ANR1H2NR1H3HTT
SCHEMBL9829823 0.79 HSD11B1 (0.62) HSD11B1TRPA1AHR
SCHEMBL9830814 0.79 HSD11B1 (0.54) HSD11B1NPC1RAB9ANR1H2NR1H3
SCHEMBL9832170 0.79 HSD11B1 (0.54) HSD11B1TRPA1CYP3A4CYP2D6CYP2C19
SCHEMBL9832924 0.79 HSD11B1 (0.48) HSD11B1CYP3A4CYP2D6CYP2C19KDM4E
SCHEMBL9829855 0.78 HSD11B1 (0.53) HSD11B1TRPA1
Fepitrizol SCHEMBL2107850 0.78 USP1 (0.47) NPC1RAB9ANR1H2NR1H3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0185256-B1 TRIAZOLE DERIVATES, THEIR PREPARATION AND THEIR USE AS PESTICIDES CIBA-GEIGY AG (CH) 1991-01-30 EP claimed
EP-0185256-A2 Triazole derivates, their preparation and their use as pesticides CIBA-GEIGY AG (CH) 1986-06-25 EP claimed
EP-0185256-B1 TRIAZOLE DERIVATES, THEIR PREPARATION AND THEIR USE AS PESTICIDES CIBA-GEIGY AG (CH) 1991-01-30 EP disclosed
US-4788210-A PESTICIDES HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed