SCHEMBL9830188

SCHEMBL9830188

Cc1cc(N(C)C)nc2ccc(Br)cc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.42
RXFP1 Q9HBX9 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MCHR1 Q99705 1/20 0.41
TP53BP1 Q12888 1/20 0.41
HTT P42858 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MPO P05164 1/20 0.41
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
BCHE P06276 2/20 0.39
ACHE P22303 2/20 0.39
GRIN1 Q05586 2/20 0.39
GRIN2A Q12879 2/20 0.39
EGFR P00533 1/20 0.39
PRNP P04156 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30048942 0.78 CYP1A2 (0.57) CASP3RXFP1CYP1A2CYP2D6CYP2C9
SCHEMBL15724648 0.78 CYP1A2 (0.57) CASP3RXFP1CYP1A2CYP2D6CYP2C9
SCHEMBL23110453 0.78 ESR1 (0.38) CASP3RXFP1CYP1A2CYP2D6CYP2C9
SCHEMBL9828594 0.77 TP53BP1 (0.45) MCHR1TP53BP1ALDH1A1KDM4EGAA
SCHEMBL6489480 0.77 CYP1A2 (0.60) CYP1A2CYP2D6CYP2C19ALDH1A1KDM4E
SCHEMBL1223950 0.75 CYP2C19 (0.62) CASP3RXFP1CYP1A2CYP2D6CYP2C9
SCHEMBL1500224 0.73 NCF1 (0.55) CYP1A2CYP2C19MCHR1HTTALDH1A1
SCHEMBL16478049 0.72 DHODH (0.51) RXFP1ALDH1A1GAANPC1
SCHEMBL1224169 0.72 L3MBTL1 (0.60) CASP3RXFP1CYP1A2CYP2D6CYP2C9
SCHEMBL5239938 0.71 ERAP1 (0.36) CYP1A2CYP2D6CYP2C19TP53BP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0096214-B1 ANTIBACTERIAL PYRIMIDINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-02-27 EP disclosed
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US disclosed
EP-0096214-A1 Antibacterial pyrimidine compounds THE WELLCOME FOUNDATION LIMITED (GB) 1983-12-21 EP disclosed