SCHEMBL9830386

SCHEMBL9830386

COc1cc(Cc2cnc(N)nc2N)ccc1N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.82
HTT P42858 1/20 0.82
MEN1 O00255 1/20 0.71
SLC22A1 O15245 1/20 0.71
ALDH1A1 P00352 1/20 0.71
CYP3A4 P08684 1/20 0.71
TSHR P16473 1/20 0.71
NFKB1 P19838 1/20 0.71
CYP2C19 P33261 1/20 0.71
BLM P54132 1/20 0.71
KMT2A Q03164 1/20 0.71
HSD17B10 Q99714 1/20 0.71
CSF1R P07333 2/20 0.68
NTRK2 Q16620 2/20 0.68
NTRK1 P04629 1/20 0.68
NTRK3 Q16288 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diaveridine SCHEMBL29527560 0.90 DHFR (1.00) DHFRHTTCSF1RNTRK2NTRK1
Diaveridine SCHEMBL93896 0.90 DHFR (1.00) DHFRHTTCSF1RNTRK2NTRK1
SCHEMBL9654048 0.86 DHFR (0.78) DHFRHTTMEN1SLC22A1ALDH1A1
Bromide SCHEMBL10488914 0.85 DHFR (0.76) DHFRHTTMEN1SLC22A1ALDH1A1
Hydrochloric Acid SCHEMBL11391196 0.85 DHFR (0.76) DHFRHTTMEN1SLC22A1ALDH1A1
SCHEMBL10488908 0.85 DHFR (0.85) DHFRHTTCSF1RNTRK2NTRK1
SCHEMBL11595225 0.84 DHFR (0.77) DHFRHTTMEN1SLC22A1ALDH1A1
SCHEMBL11546389 0.84 DHFR (0.74) DHFRHTTMEN1SLC22A1ALDH1A1
Aditeren SCHEMBL1230789 0.84 DHFR (0.81) DHFRHTTMEN1SLC22A1ALDH1A1
SCHEMBL9657245 0.84 DHFR (0.78) DHFRHTTCSF1RNTRK2NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0096214-B1 ANTIBACTERIAL PYRIMIDINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-02-27 EP disclosed
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US disclosed
EP-0096214-A1 Antibacterial pyrimidine compounds THE WELLCOME FOUNDATION LIMITED (GB) 1983-12-21 EP disclosed