SCHEMBL9830388

SCHEMBL9830388

COC(=O)c1cccc(Cl)c1NS(=O)(=O)c1nc2ncc(C)cn2n1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
LCK P06239 1/20 0.38
MAPT P10636 2/20 0.37
FFAR4 Q5NUL3 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SLC40A1 Q9NP59 1/20 0.35
F2 P00734 1/20 0.34
KMT2A Q03164 3/20 0.34
SCN9A Q15858 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 2/20 0.34
PTGS2 P35354 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832928 0.92 AURKB (0.39) LMNAMAPK1MAPTKDM4EALDH1A1
SCHEMBL9831611 0.91 MAPT (0.35) LCKMAPTKDM4EALDH1A1NPC1
SCHEMBL9832148 0.90 FFAR4 (0.37) LMNAMAPK1LCKMAPTFFAR4
SCHEMBL9832083 0.90 ACLY (0.39) LMNAMAPTKMT2AMEN1PTGS2
SCHEMBL9832129 0.88 MAPT (0.36) LMNAMAPK1MAPTFFAR4ALDH1A1
SCHEMBL9831382 0.88 MAPT (0.36) LMNAMAPK1LCKMAPTALDH1A1
SCHEMBL9830333 0.88 KMT2A (0.37) LMNAMAPK1MAPTFFAR4KDM4E
SCHEMBL9830515 0.88 SLC40A1 (0.35) SLC40A1KMT2A
SCHEMBL9832418 0.86 ACLY (0.40) LMNAMAPK1LCKMAPTFFAR4
SCHEMBL9831264 0.86 ABL1 (0.36) LMNAMAPTFFAR4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed