SCHEMBL9830832

SCHEMBL9830832

CCn1nc(-c2ccccc2C(F)(F)F)nc1-c1ccccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 9/20 0.44
CYP1A2 P05177 5/20 0.39
CYP3A4 P08684 3/20 0.39
HSD17B10 Q99714 3/20 0.39
ALDH1A1 P00352 3/20 0.39
CYP2C19 P33261 3/20 0.39
NR1H3 Q13133 2/20 0.39
TSHR P16473 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
ALOX15 P16050 1/20 0.39
MAPK1 P28482 1/20 0.39
HIF1A Q16665 1/20 0.39
NR1H2 P55055 1/20 0.39
KCNN4 O15554 1/20 0.39
CYP2D6 P10635 3/20 0.38
CYP2C9 P11712 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
RECQL P46063 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9829646 0.95 HSD11B1 (0.47) HSD11B1HSD17B10ALDH1A1NR1H3NR1H2
SCHEMBL9829810 0.86 HSD11B1 (0.54) HSD11B1CYP1A2CYP3A4HSD17B10ALDH1A1
SCHEMBL9830637 0.83 HSD11B1 (0.54) HSD11B1NR1H3NR1H2
SCHEMBL9829686 0.82 HSD11B1 (0.50) HSD11B1CYP1A2CYP3A4HSD17B10ALDH1A1
SCHEMBL9830362 0.82 HSD11B1 (0.45) HSD11B1NR1H3NR1H2KDM4E
SCHEMBL9829855 0.77 HSD11B1 (0.53) HSD11B1KCNN4
SCHEMBL9831536 0.76 HSD11B1 (0.55) HSD11B1CYP1A2CYP3A4HSD17B10ALDH1A1
SCHEMBL9830317 0.73 HSD11B1 (0.55) HSD11B1
SCHEMBL9830541 0.73 HSD11B1 (0.58) HSD11B1CYP1A2CYP3A4HSD17B10ALDH1A1
SCHEMBL9830794 0.72 HSD11B1 (0.53) HSD11B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4788210-A PESTICIDES HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US claimed
EP-0185256-B1 TRIAZOLE DERIVATES, THEIR PREPARATION AND THEIR USE AS PESTICIDES CIBA-GEIGY AG (CH) 1991-01-30 EP disclosed
US-4788210-A PESTICIDES HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed
EP-0185256-A2 Triazole derivates, their preparation and their use as pesticides CIBA-GEIGY AG (CH) 1986-06-25 EP disclosed