SCHEMBL9830968

SCHEMBL9830968

Cc1cc(C)c2cccc(Cl)c2n1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 4/20 0.69
KDM4E B2RXH2 2/20 0.62
TDP1 Q9NUW8 1/20 0.62
CRHR1 P34998 4/20 0.62
L3MBTL1 Q9Y468 2/20 0.50
MAPT P10636 1/20 0.50
CYP1A2 P05177 1/20 0.50
PARP1 P09874 1/20 0.49
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.46
ALDH1A1 P00352 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.44
TP53 P04637 1/20 0.42
ACHE P22303 1/20 0.42
CCR1 P32246 1/20 0.42
CCR8 P51685 1/20 0.42
CYP3A4 P08684 1/20 0.42
CD38 P28907 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063558 0.86 NR4A2 (0.71) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL8966258 0.82 KDM4E (0.69) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL438980 0.81 NR4A2 (1.00) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL1026984 0.81 NR4A2 (0.65) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL1715255 0.79 KDM4E (0.61) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL24425989 0.79 NR4A2 (0.61) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL11570729 0.79 NR4A2 (0.61) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL28046875 0.78 NR4A2 (0.59) NR4A2KDM4ECRHR1L3MBTL1MAPT
SCHEMBL6726554 0.77 CRHR1 (1.00) NR4A2KDM4ETDP1CRHR1L3MBTL1
SCHEMBL11585401 0.77 KDM4E (1.00) NR4A2KDM4ETDP1CRHR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0096214-B1 ANTIBACTERIAL PYRIMIDINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-02-27 EP disclosed
US-4587341-A BACTERICIDES BURROUGHS WELLCOME CO. (US) 1986-05-06 US disclosed
EP-0096214-A1 Antibacterial pyrimidine compounds THE WELLCOME FOUNDATION LIMITED (GB) 1983-12-21 EP disclosed