SCHEMBL9832040

SCHEMBL9832040

CC(C)(C)NC(=O)C(C#N)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccccc1-2

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 0.43
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
RAB9A P51151 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPT P10636 6/20 0.39
KMT2A Q03164 1/20 0.39
THRB P10828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833371 0.92 MAPT (0.40) TP53RAB9AL3MBTL1MAPTKMT2A
SCHEMBL9522614 0.88 MAPT (0.43) TP53PTGS1PTGS2RAB9AL3MBTL1
SCHEMBL9522928 0.87 TP53 (0.42) TP53PTGS1PTGS2RAB9AL3MBTL1
SCHEMBL8111901 0.87 TP53 (0.42) TP53PTGS1PTGS2RAB9AL3MBTL1
SCHEMBL9832793 0.87 TP53 (0.46) TP53PTGS1PTGS2RAB9AL3MBTL1
SCHEMBL9526191 0.86 TP53 (0.42) TP53PTGS1PTGS2RAB9AL3MBTL1
SCHEMBL9316737 0.86 TP53 (0.49) TP53PTGS1PTGS2RAB9AL3MBTL1
SCHEMBL9836400 0.85 MAPT (0.46) TP53RAB9AL3MBTL1MAPTKMT2A
SCHEMBL9833687 0.85 TP53 (0.41) TP53RAB9AL3MBTL1MAPTKMT2A
SCHEMBL9834988 0.85 TP53 (0.41) TP53PTGS1PTGS2RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed