SCHEMBL9832793

SCHEMBL9832793

N#CC(C(=O)O)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccccc1-2

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.46
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
THRB P10828 1/20 0.41
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 4/20 0.39
KMT2A Q03164 1/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8113736 0.92 TP53 (0.45) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9339764 0.92 TP53 (0.45) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL8111901 0.88 TP53 (0.42) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9522928 0.88 TP53 (0.42) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9316737 0.87 TP53 (0.49) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9832040 0.87 TP53 (0.43) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9834217 0.87 TP53 (0.43) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9834215 0.87 TP53 (0.41) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9316088 0.85 TP53 (0.44) TP53PTGS1PTGS2THRBRAB9A
SCHEMBL9526191 0.85 TP53 (0.42) TP53PTGS1PTGS2THRBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed