SCHEMBL9832146

SCHEMBL9832146

Nc1n[nH]cc1C(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 1/20 0.50
CES2 O00748 1/20 0.50
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
MAPT P10636 1/20 0.48
ADORA1 P30542 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TLR7 Q9NYK1 2/20 0.46
CNR2 P34972 2/20 0.46
PTGS1 P23219 4/20 0.45
NPSR1 Q6W5P4 1/20 0.45
VNN1 O95497 4/20 0.44
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831962 0.82 PARP1 (0.47) CES2MEN1ALDH1A1KMT2ACCNA2
SCHEMBL30877071 0.82 CES2 (0.41) CES2MEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL30877077 0.82 CES2 (0.41) CES2MEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL9832118 0.79 POLB (0.51) ALDH1A1MAPTKMT2ANPSR1VNN1
SCHEMBL3982930 0.78 MAPT (0.52) MEN1ALDH1A1MAPTADORA1KMT2A
SCHEMBL5347968 0.76 PTGS1 (0.59) SRD5A2CES2MEN1ALDH1A1CYP1A2
SCHEMBL1237189 0.75 SRD5A2 (0.79) SRD5A2CES2MEN1ALDH1A1CYP1A2
SCHEMBL2079912 0.73 VNN1 (0.51) SRD5A2CES2MEN1ALDH1A1CYP1A2
SCHEMBL4710822 0.73 MEN1 (0.54) SRD5A2CES2MEN1ALDH1A1CYP1A2
SCHEMBL15608381 0.72 MEN1 (0.56) SRD5A2CES2MEN1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129846-B1 (3-AMINO-1H-PYRAZOL-4-YL)(ARYL)METHANONES AMERICAN CYANAMID COMPANY (US) 1991-05-08 EP claimed
EP-0129846-A2 (3-Amino-1H-pyrazol-4-yl)(aryl)methanones AMERICAN CYANAMID COMPANY (US) 1985-01-02 EP claimed