SCHEMBL9832367

SCHEMBL9832367

COC(=O)c1ccc(C)c(C)c1NS(=O)(=O)c1nc2nccc(C)n2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
SMN1; SMN2 Q16637 5/20 0.45
KMT2A Q03164 3/20 0.45
RECQL P46063 1/20 0.45
L3MBTL1 Q9Y468 3/20 0.41
NPC1 O15118 5/20 0.40
RAB9A P51151 5/20 0.40
PKM P14618 1/20 0.40
RXFP1 Q9HBX9 2/20 0.40
MEN1 O00255 2/20 0.39
TSHR P16473 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.38
MAPK1 P28482 2/20 0.37
POLB P06746 2/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
SLC40A1 Q9NP59 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9830969 0.91 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9832400 0.90 L3MBTL1 (0.40) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9830619 0.90 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9832696 0.89 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9832594 0.88 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9831673 0.87 L3MBTL1 (0.50) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9832066 0.86 TSHR (0.55) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9831239 0.85 L3MBTL1 (0.45) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9832043 0.83 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1
SCHEMBL9831860 0.83 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2KMT2ARECQLL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP claimed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP claimed
EP-0142152-B1 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1991-03-20 EP disclosed
EP-0413020-A1 PYRAZOLOTRIAZOLES AND PROCESSES FOR THEIR FORMATION EASTMAN KODAK COMPANY (US) 1991-02-20 EP disclosed
US-4977269-A ANHYDROUS REACTION WITH CARBOXYLIC ACID, ANHYDRIDE OR ACYL HALIDE WITH LEWIS ACID CATALYST EASTMAN KODAK COMPANY (US) 1990-12-11 US disclosed
WO-1990010004-A1 PYRAZOLOTRIAZOLES AND PROCESSES FOR THEIR FORMATION EASTMAN KODAK COMPANY (US) 1990-09-07 WO disclosed
US-4914209-A PHOTOGRAPHIC COUPLERS EASTMAN KODAK COMPANY (US) 1990-04-03 US disclosed
EP-0330137-A1 Intermediate compounds for the preparation of 1,2,4-triazolo [1,5-a]pyrimidine-2-sulfonamides DowElanco (US) 1989-08-30 EP disclosed
US-4755212-A Novel substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonamides and compositions and method for inhibiting pollen formation in corn THE DOW CHEMICAL COMPANY (US) 1988-07-05 US disclosed
US-4741764-A SUPPRESSION OF NITRIFICATION OF AMMONIUM NITROGEN IN THE SOIL THE DOW CHEMICAL COMPANY (US) 1988-05-03 US disclosed
US-4740233-A Substituted 1,2,4-triazolo[1,5-a]-pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1988-04-26 US disclosed
EP-0142152-A2 Novel substituted 1,2,4-triazolo- [1,5-a] pyrimidine-2-sulfonamides and compositions and methods of controlling undesired vegetation and suppressing the nitrification of ammonium nitrogen in soil THE DOW CHEMICAL COMPANY (US) 1985-05-22 EP disclosed