SCHEMBL9832621

SCHEMBL9832621

CC(=O)N1c2ccccc2Sc2nccnc21

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 1/20 0.61
HDAC6 Q9UBN7 1/20 0.49
BCHE P06276 15/20 0.49
POLB P06746 1/20 0.46
ATM Q13315 1/20 0.46
ACHE P22303 3/20 0.45
SNCA P37840 1/20 0.45
GLA P06280 1/20 0.44
ALOX15 P16050 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832954 0.85 BCHE (0.64) NOX1HDAC6BCHEPOLBACHE
SCHEMBL18612766 0.84 NOX1 (0.68) NOX1BCHEPOLBATMACHE
SCHEMBL25388003 0.84 NOX1 (0.68) NOX1HDAC6BCHEPOLBATM
SCHEMBL6747160 0.80 NOX1 (0.37) NOX1HDAC6SNCA
SCHEMBL9830999 0.79 SNCA (0.54) NOX1BCHEACHESNCAALOX15
SCHEMBL30198410 0.77 NOX1 (1.00) NOX1BCHEPOLBATMACHE
SCHEMBL341905 0.77 NOX1 (1.00) NOX1BCHEPOLBATMACHE
SCHEMBL9832554 0.76 MAOA (0.55) NOX1HDAC6POLBSMN1; SMN2GAA
SCHEMBL9832223 0.74 HDAC6 (0.59) HDAC6MAPT
SCHEMBL12165688 0.73 HDAC6 (0.43) NOX1HDAC6BCHESMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0140709-B1 5-LIPOXYGENASE INHIBITORS MERCK FROSST CANADA INC. (CA) 1991-04-03 EP disclosed
US-4634766-A LIPOXYGENASE INHIBITORS MERCK FROSST CANADA, INC. (CA) 1987-01-06 US disclosed
EP-0140709-A2 5-Lipoxygenase inhibitors MERCK FROSST CANADA INC. (CA) 1985-05-08 EP disclosed