SCHEMBL9833015

SCHEMBL9833015

COc1ccc(CSc2c(CO)cccc2[N+](=O)[O-])cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.48
PTPN1 P18031 1/20 0.47
ALDH1A1 P00352 6/20 0.44
NPC1 O15118 3/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
RAB9A P51151 2/20 0.42
MAPK1 P28482 2/20 0.42
DCTPP1 Q9H773 1/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 3/20 0.42
HTT P42858 1/20 0.42
NCOA1 Q15788 1/20 0.42
NCOA3 Q9Y6Q9 1/20 0.42
MAPT P10636 3/20 0.41
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
SLC29A1 Q99808 1/20 0.40
CA2 P00918 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833207 0.82 HPGD (0.53) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL10831867 0.81 HPGD (0.55) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL8996846 0.79 SMN1; SMN2 (0.51) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL7398084 0.76 ALDH1A1 (0.49) HPGDALDH1A1NPC1SMN1; SMN2RAB9A
SCHEMBL9831716 0.74 CACNA1C (0.69) HPGDALDH1A1SMN1; SMN2MAPK1KMT2A
SCHEMBL5795803 0.72 KMT2A (0.71) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL3825495 0.72 PTPN1 (0.67) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL5201436 0.71 ALDH1A1 (0.47) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL31347487 0.71 ALDH1A1 (0.47) HPGDPTPN1ALDH1A1NPC1SMN1; SMN2
SCHEMBL8349572 0.70 ALDH1A1 (0.44) HPGDALDH1A1NPC1SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0163238-B1 SUBSTITUTED AND BRIDGED PYRIDINES USEFUL AS PHARMACEUTICAL AGENTS MERCK & CO. INC. (US) 1991-07-24 EP disclosed
US-4579851-A HYPOTENSIVE, ANTIARRHYTHMIA AGENTS MERCK & CO., INC. (US) 1986-04-01 US disclosed
EP-0163238-A2 Substituted and bridged pyridines useful as pharmaceutical agents MERCK & CO. INC. (US) 1985-12-04 EP disclosed